SCHEMBL748950

SCHEMBL748950

CC1C2CCN1CC(Oc1cnc(-c3cnc4[nH]ccc4c3)cn1)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.44
CHRNB2 P17787 2/20 0.44
CHRNB4 P30926 2/20 0.44
CHRNA3 P32297 2/20 0.44
CHRNA4 P43681 2/20 0.44
LRRK2 Q5S007 1/20 0.38
PIK3CD O00329 3/20 0.37
MTOR P42345 1/20 0.37
BRD4 O60885 1/20 0.36
AXL P30530 2/20 0.36
CDK8 P49336 2/20 0.36
FEN1 P39748 2/20 0.36
ALOX5AP P20292 1/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36
PIK3CA P42336 2/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
PRKCZ Q05513 1/20 0.35
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL747272 0.79 PIK3CA (0.41) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL747739 0.71 PIK3CD (0.38) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2671996 0.71 MTOR (0.42) LRRK2PIK3CDMTORBRD4AXL
SCHEMBL746345 0.68 PRKCZ (0.43) PIK3CDMTORBRD4AXLCDK8
SCHEMBL2672158 0.67 MTOR (0.41) CHRNA7LRRK2PIK3CDMTORBRD4
SCHEMBL2672618 0.67 CDK8 (0.45) LRRK2PIK3CDMTORBRD4AXL
SCHEMBL743968 0.66 CHRNA7 (0.53) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL743970 0.66 PRKCZ (0.46) PIK3CDBRD4AXLCDK8PIK3CA
SCHEMBL18857740 0.66 CHRNA7 (0.65) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL3390939 0.66 CHRNA7 (0.65) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431368-A1 CNS active fused bicycloheterocycle substituted azabicyclic alkane derivatives Abbott Laboratories (US) 2012-03-21 EP disclosed