SCHEMBL7490272

SCHEMBL7490272

CC(C)=N/N=C1\NC(=O)C(CC(=O)Nc2ccc(C)cc2)S1

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.70
KDM4E B2RXH2 2/20 0.70
MAPT P10636 7/20 0.68
GAA P10253 2/20 0.67
ALDH1A1 P00352 1/20 0.66
MEN1 O00255 6/20 0.62
KMT2A Q03164 6/20 0.62
HTT P42858 1/20 0.62
RECQL P46063 1/20 0.62
POLB P06746 3/20 0.61
XBP1 P17861 1/20 0.61
HPGD P15428 1/20 0.59
TDP1 Q9NUW8 1/20 0.54
LMNA P02545 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7490274 1.00 L3MBTL1 (0.70) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7494297 0.91 MAPT (0.60) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7494293 0.91 MAPT (0.60) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7491013 0.90 MAPT (0.59) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7501258 0.90 MAPT (0.72) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7491005 0.90 MAPT (0.59) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7501266 0.90 MAPT (0.72) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7488228 0.90 MAPT (0.63) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL3500377 0.90 MAPT (0.63) L3MBTL1KDM4EMAPTGAAALDH1A1
SCHEMBL7490971 0.90 MAPT (0.63) L3MBTL1KDM4EMAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638075-B1 THIAZOLE OR IMIDAZOLE DERIVATIVES AS MAILLARD REACTION INHIBITORS OTSUKA PHARMA CO LTD (JP) 2002-01-16 EP disclosed
EP-0638075-A1 THIAZOLE OR IMIDAZOLE DERIVATIVES AS MAILLARD REACTION INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-02-15 EP disclosed
WO-1994019335-A1 THIAZOLE OR IMIDAZOLE DERIVATIVES AS MAILLARD REACTION INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-09-01 WO disclosed