SCHEMBL7490398

SCHEMBL7490398

O=C(O)c1cnc2ccc(Br)cc2c1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
TSHR P16473 1/20 0.50
DHODH Q02127 4/20 0.49
MALT1 Q9UDY8 1/20 0.45
RXFP1 Q9HBX9 6/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.43
KDM4E B2RXH2 4/20 0.43
PPARG P37231 3/20 0.43
NCOR2 Q9Y618 3/20 0.43
ALDH1A1 P00352 3/20 0.43
POLB P06746 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
RECQL P46063 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ESR1 P03372 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17241522 0.88 HTT (0.50) HTTTSHRDHODHMALT1RXFP1
SCHEMBL25311292 0.88 DHODH (0.43) HTTTSHRDHODHRXFP1MEN1
SCHEMBL529214 0.86 HTT (0.63) HTTTSHRDHODHMALT1RXFP1
SCHEMBL2725311 0.86 HTT (0.49) HTTTSHRDHODHMALT1RXFP1
Hydrochloric Acid SCHEMBL25311682 0.86 DHODH (0.42) HTTTSHRDHODHRXFP1MEN1
SCHEMBL2721434 0.84 LMNA (0.58) TSHRDHODHMEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL9872122 0.83 LMNA (0.60) TSHRDHODHMEN1KMT2ALMNA
SCHEMBL741418 0.83 HTT (0.55) HTTTSHRDHODHRXFP1MEN1
SCHEMBL403348 0.82 TSHR (0.66) HTTTSHRMALT1RXFP1KDM4E
SCHEMBL10282056 0.82 HTT (0.49) HTTTSHRDHODHMALT1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255692-A Imidazo [4,5-c ] quinolin-2-one compounds and their use in treating cancer 阿斯利康(瑞典)有限公司 2016-12-21 CN disclosed
CN-105859684-A Fused ring compound and preparation method, application and intermediate compound thereof 四川赛诺唯新生物技术有限公司 2016-08-17 CN disclosed
CN-103476755-B Compounds and methods for CLANOTECH AB (SE) 2015-08-26 CN disclosed
CN-103044446-A Heterocycle quinoline derivatives as well as medicinal salts, preparation method and medicinal application thereof SHANGHAI HENGRUI PHARM CO LTD 2013-04-17 CN disclosed
WO-2008119771-A2 QUINOLINE-S-CARBOXYLIC ACID DERIVATIVES AS TYROSINE KINASE INHIBITORS CLANOTECH AB (SE) 2008-10-09 WO disclosed
CN-1097459-C Diazepino-indoles as phosphodiesterase IV inhibitors JOUVEINAL INST RECH (FR) 2003-01-01 CN disclosed
EP-0785789-B1 DIAZEPINO-INDOLES AS PHOSPHODIESTERASE IV INHIBITORS PFIZER (FR) 2002-09-11 EP disclosed
CN-1160352-A Diaza * -oxindoles as phosphodiesterase IV inhibitors JOUVEINAL INST RECH (FR) 1997-09-24 CN disclosed
EP-0785789-A1 DIAZEPINO-INDOLES AS PHOSPHODIESTERASE IV INHIBITORS INSTITUT DE RECHERCHE JOUVEINAL (I.R.J) (FR) 1997-07-30 EP disclosed
WO-1996011690-A1 DIAZEPINO-INDOLES AS PHOSPHODIESTERASE IV INHIBITORS INSTITUT DE RECHERCHE JOUVEINAL (FR) 1996-04-25 WO disclosed