SCHEMBL7490457

SCHEMBL7490457

Cc1[nH]c2ccccc2c1C=C1C(=O)NN=C1c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
KDR P35968 3/20 0.45
ALK Q9UM73 1/20 0.43
MEN1 O00255 3/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.40
PSMD14 O00487 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PLK4 O00444 1/20 0.39
FLT3 P36888 1/20 0.39
GAA P10253 1/20 0.39
TDO2 P48775 1/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
MCL1 Q07820 1/20 0.38
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7489879 0.78 GAA (0.39) KDRMEN1MAPTKMT2ALMNA
SCHEMBL6089157 0.78 NTRK1 (0.49) KDRALKMEN1MAPTKMT2A
SCHEMBL6089153 0.78 NTRK1 (0.49) KDRALKMEN1MAPTKMT2A
SCHEMBL6089787 0.77 KDR (0.42) CYP11B1CYP11B2KDRALKMEN1
SCHEMBL6089795 0.77 KDR (0.42) CYP11B1CYP11B2KDRALKMEN1
SCHEMBL7489423 0.77 GAA (0.45) MEN1MAPTKMT2ALMNAALDH1A1
SCHEMBL6090995 0.76 KDR (0.49) KDRALKKMT2ALMNAALDH1A1
SCHEMBL6090988 0.76 KDR (0.49) KDRALKKMT2ALMNAALDH1A1
SCHEMBL6092766 0.76 CYP19A1 (0.49) KDRALKMAPTLMNAALDH1A1
SCHEMBL6092761 0.76 CYP19A1 (0.49) KDRALKMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP disclosed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed