SCHEMBL6089795

SCHEMBL6089795

CCOC(=O)c1c(C=C2C(=O)NN=C2c2cccnc2)[nH]c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.42
ALK Q9UM73 2/20 0.41
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
ABL1 P00519 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
FLT3 P36888 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6089787 1.00 KDR (0.42) KDRALKMMP2MMP13MMP14
SCHEMBL6089402 0.87 KDR (0.52) KDRALKABL1RETPDGFRB
SCHEMBL6089417 0.87 KDR (0.52) KDRALKABL1RETPDGFRB
SCHEMBL6089380 0.84 ALK (0.56) KDRALKMMP2MMP13MMP14
SCHEMBL6089385 0.84 ALK (0.56) KDRALKMMP2MMP13MMP14
SCHEMBL6088717 0.82 ABL1 (0.40) KDRALKABL1RETPDGFRB
SCHEMBL6088711 0.82 ABL1 (0.40) KDRALKABL1RETPDGFRB
SCHEMBL6093374 0.82 ALK (0.41) KDRALKMMP2MMP13MMP14
SCHEMBL6093367 0.82 ALK (0.41) KDRALKMMP2MMP13MMP14
SCHEMBL6088582 0.81 NPSR1 (0.44) ALKABL1RETPDGFRBFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed