SCHEMBL7495262

SCHEMBL7495262

O=C(Nc1ccc([N+](=O)[O-])cc1O)Nc1ccccc1Oc1ccccc1.O=C(Nc1ccccc1Br)Nc1cccc(Cl)c1O

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 12/20 0.66
CXCR1 P25024 8/20 0.66
MEN1 O00255 4/20 0.66
KMT2A Q03164 4/20 0.66
TDP1 Q9NUW8 2/20 0.66
HDAC6 Q9UBN7 1/20 0.66
MAPT P10636 4/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
NPC1 O15118 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
PYGL P06737 1/20 0.42
PYGM P11217 1/20 0.42
RORC P51449 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7491012 0.88 CXCR2 (0.70) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL3708973 0.87 CXCR1 (0.67) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL5595225 0.81 MEN1 (0.60) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL29733649 0.81 CXCR2 (1.00) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL29493172 0.81 CXCR2 (1.00) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL1110610 0.81 CXCR2 (1.00) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL6921874 0.81 CXCR2 (1.00) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL7622098 0.76 MAPT (0.61) MEN1KMT2ATDP1MAPTALDH1A1
SCHEMBL3706835 0.76 KMT2A (0.74) CXCR2CXCR1MEN1KMT2ATDP1
SCHEMBL7493083 0.76 CXCR2 (0.74) CXCR2CXCR1MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0896531-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-10-30 EP disclosed
EP-0896531-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-17 EP disclosed
WO-1997029743-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-21 WO disclosed