SCHEMBL7496263

SCHEMBL7496263

NC(=O)NCC12CN(c3c(F)cc4c(=O)c(OC(=O)O)cn(C5CC5)c4c3F)CC1CCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.40
ALDH1A1 P00352 5/20 0.37
POLB P06746 3/20 0.37
OPRM1 P35372 2/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
OPRD1 P41143 1/20 0.37
TOP2A P11388 2/20 0.36
TOP2B Q02880 2/20 0.36
KDM4E B2RXH2 5/20 0.36
HPGD P15428 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
HSD17B10 Q99714 2/20 0.36
PRKD3 O94806 1/20 0.36
ALOX15 P16050 1/20 0.36
CLK2 P49760 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
ADRB2 P07550 1/20 0.35
LMNA P02545 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499642 0.93 ALDH1A1 (0.46) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7496259 0.90 KCNH2 (0.51) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7495789 0.90 KCNH2 (0.39) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7495693 0.90 KCNH2 (0.46) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7496654 0.90 KCNH2 (0.37) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7494369 0.90 KCNH2 (0.37) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7501610 0.90 KCNH2 (0.37) KCNH2ALDH1A1POLBOPRM1CHRM2
SCHEMBL7497800 0.90 KCNH2 (0.39) KCNH2ALDH1A1POLBOPRM1CHRM2
Hydrochloric Acid SCHEMBL7503689 0.90 KCNH2 (0.40) KCNH2ALDH1A1POLBOPRM1CHRM2
Hydrochloric Acid SCHEMBL7501440 0.89 KCNH2 (0.46) KCNH2ALDH1A1POLBOPRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944385-B1 USE OF 7-(1-AMINOMETHYL-2-OXA-7-AZA-BICYCLO 3.3.0]OCT-7-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDONE CARBOXYLIC ACID DERIVATIVES FOR TREATING HELICOBACTER PYLORI INFECTIONS AND THE GASTRODUODENAL DISEASES ASSOCIATED THEREWITH BAYER AG (DE) 2002-10-16 EP disclosed