SCHEMBL7497633

SCHEMBL7497633

CC(=O)N1c2ccccc2N(Cc2ccccc2)C(=O)[C@H]2CCC[C@H]21

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.55
ALDH1A1 P00352 4/20 0.55
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.53
POLB P06746 1/20 0.53
HDAC6 Q9UBN7 2/20 0.45
MT-CO2 P00403 1/20 0.44
ALOX5 P09917 1/20 0.44
MAPK1 P28482 1/20 0.44
CREBBP Q92793 1/20 0.43
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7497627 1.00 BRD4 (0.55) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7497359 0.87 ALDH1A1 (0.53) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7497354 0.87 ALDH1A1 (0.53) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7502533 0.87 ALDH1A1 (0.48) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7502537 0.87 ALDH1A1 (0.48) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7498069 0.86 ALDH1A1 (0.56) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7498239 0.86 ALDH1A1 (0.52) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7500262 0.86 ALDH1A1 (0.52) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7501263 0.86 ALDH1A1 (0.52) BRD4ALDH1A1KMT2AMEN1POLB
SCHEMBL7495825 0.86 ALDH1A1 (0.52) BRD4ALDH1A1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed