SCHEMBL7497657

SCHEMBL7497657

Clc1cccc(Nc2nc[nH]c3nc4ccccc4c2-3)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.54
FADS1 O60427 4/20 0.54
PDE5A O76074 3/20 0.54
ABCG2 Q9UNQ0 2/20 0.54
LCK P06239 1/20 0.53
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
BRAF P15056 1/20 0.48
ABL1 P00519 1/20 0.46
ABL2 P42684 1/20 0.46
TTBK1 Q5TCY1 1/20 0.46
TTBK2 Q6IQ55 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7499724 0.99 EGFR (0.55) EGFRFADS1PDE5AABCG2LCK
SCHEMBL7216427 0.87 NPY5R (0.47) EGFRPDE5AABCG2KDM4ESMN1; SMN2
SCHEMBL7222295 0.85 EGFR (0.54) EGFRABCG2BRAF
Hydrochloric Acid SCHEMBL7218002 0.84 EGFR (0.53) EGFRABCG2BRAF
SCHEMBL19261422 0.74 PDE5A (0.70) EGFRFADS1PDE5AABCG2LCK
SCHEMBL4740823 0.73 PDE5A (0.72) EGFRFADS1PDE5AABCG2LCK
SCHEMBL2389719 0.72 GUSB (0.43) KDM4ESMN1; SMN2NPC1RAB9AMEN1
SCHEMBL17432159 0.72 MEN1 (0.79) EGFRFADS1PDE5AABCG2LCK
SCHEMBL7494318 0.71 EGFR (0.49) EGFRFADS1PDE5AABCG2LCK
Hydrochloric Acid SCHEMBL7218019 0.71 GUSB (0.42) KDM4ESMN1; SMN2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836605-B1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 2002-02-06 EP disclosed
US-6140332-A Pyrrolopyrimidines and processes for the preparation thereof NOVARTIS AG (CH) 2000-10-31 US disclosed
EP-0836605-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF Novartis AG (CH) 1998-04-22 EP disclosed
WO-1997002266-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 1997-01-23 WO disclosed