SCHEMBL7498447

SCHEMBL7498447

O[C@H](CNCc1ccc(F)cc1F)COc1ccc(-c2onc3cc(F)ccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
ADRB1 P08588 3/20 0.39
ADRB3 P13945 3/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ROCK2 O75116 1/20 0.38
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35
KDM1A O60341 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
HPGD P15428 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CDK4 P11802 1/20 0.34
CDK2 P24941 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1384566 0.89 NPC1 (0.57) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL1384570 0.89 NPC1 (0.57) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL7496503 0.87 NPC1 (0.40) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL7496514 0.87 NPC1 (0.40) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL7493743 0.87 NPC1 (0.48) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL7487764 0.87 MEN1 (0.51) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL7499279 0.85 NPC1 (0.51) NPC1MEN1KMT2A
SCHEMBL1384330 0.84 NPC1 (0.41) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL1384333 0.84 NPC1 (0.41) NPC1ADRB1ADRB3MEN1KMT2A
SCHEMBL1384202 0.84 NPC1 (0.45) NPC1ADRB1ADRB3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed