SCHEMBL7498563

SCHEMBL7498563

COc1ccc(N2CCc3c2c2cccc(OC(F)(F)F)c2[nH]c3=O)c(C)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
MEN1 O00255 1/20 0.40
JAK2 O60674 1/20 0.40
GAA P10253 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 3/20 0.39
GRM5 P41594 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CRHR1 P34998 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAD52 P43351 1/20 0.39
PDE5A O76074 3/20 0.38
CYP1A1 P04798 2/20 0.38
CYP1B1 Q16678 2/20 0.38
TUBB4A P04350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7489265 0.91 CRHR1 (0.39) KDM4EALDH1A1CRHR1
SCHEMBL8487677 0.91 CYP1A2 (0.46) CYP1A2CYP3A4CYP2D6MEN1JAK2
SCHEMBL7490357 0.90 KDM4E (0.41) KDM4EALDH1A1CRHR1
SCHEMBL7484660 0.89 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6MEN1JAK2
SCHEMBL7496561 0.88 KDM4E (0.40) KDM4EALDH1A1CRHR1PDE5A
SCHEMBL8071575 0.87 KDM4E (0.41) KDM4EALDH1A1
SCHEMBL8481514 0.86 CYP1A2 (0.43) CYP1A2CYP3A4CYP2D6MEN1JAK2
SCHEMBL7498546 0.85 KDM4E (0.51) CYP1A2GAAKDM4EALDH1A1PDE5A
SCHEMBL7489494 0.84 KDM4E (0.40) KDM4EALDH1A1
SCHEMBL8484525 0.83 NQO2 (0.44) GAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966466-B1 PYRROLO 3,2-c]QUINOLINE DERIVATIVES CONTAINING HALOALKOXY GROUP AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF KOREA RES INST CHEM TECH (KR) 2002-07-03 EP disclosed
US-6011044-A ANTIULCER AGENTS KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2000-01-04 US disclosed