SCHEMBL7499179

SCHEMBL7499179

O=C(c1[nH]c2ncccc2c1C1=CCN2CCCC2C1)c1c(Cl)cccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.35
HTR6 P50406 1/20 0.34
OPRM1 P35372 2/20 0.33
CCR3 P51677 1/20 0.33
NUDT1 P36639 1/20 0.33
CDK9 P50750 4/20 0.33
CCNT1 O60563 3/20 0.33
HSD11B1 P28845 3/20 0.33
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
P2RX7 Q99572 1/20 0.32
CALCRL Q16602 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
RORC P51449 1/20 0.32
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499596 0.87 CCNT1 (0.39) CDK9CCNT1
SCHEMBL2063892 0.74 ELANE (0.40) HTR6RORC
SCHEMBL2063653 0.69 TMEM97 (0.47) ALKCDK9CCNT1
SCHEMBL2064415 0.68 BTK (0.35) HTR6OPRM1RORCBTK
SCHEMBL30908939 0.63 DAO (0.39) HTR6
SCHEMBL2064496 0.63 ELANE (0.38) ALDH1A1
SCHEMBL6669246 0.63 BCHE (0.46) HTR6HSD11B1GAARORC
SCHEMBL2064707 0.63 ELANE (0.43) HTR6
SCHEMBL1445398 0.62 MCHR1 (0.41) ALKOPRM1OPRD1OPRK1OPRL1
SCHEMBL7503378 0.62 CCNT1 (0.43) HTR6CDK9CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204662-A1 AZAINDOLES HAVING SEROTONIN RECEPTOR AFFINITY NPS Allelix Corp. (CA) 2002-05-15 EP disclosed
WO-2001012629-A1 AZAINDOLES HAVING SEROTONIN RECEPTOR AFFINITY NPS ALLELIX CORP. (US) 2001-02-22 WO disclosed