SCHEMBL7499341

SCHEMBL7499341

Cc1cccc(C)c1COc1cccn2c(C)c(C)nc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 1.00
CYP2C9 P11712 4/20 1.00
CYP1A2 P05177 3/20 1.00
CYP2D6 P10635 3/20 1.00
CYP2C19 P33261 2/20 1.00
ATP4A P20648 3/20 0.52
ATP4B P51164 3/20 0.52
PSEN1 P49768 1/20 0.51
PSEN2 P49810 1/20 0.51
APH1B Q8WW43 1/20 0.51
NCSTN Q92542 1/20 0.51
APH1A Q96BI3 1/20 0.51
PSENEN Q9NZ42 1/20 0.51
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
KMT2A Q03164 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
GUCY1B2 O75343 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803895 0.91 CYP3A4 (0.83) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL7216941 0.90 CYP3A4 (0.81) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL7496960 0.88 CYP3A4 (0.79) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL18801023 0.86 CYP1A2 (0.76) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL7501458 0.86 CYP3A4 (0.74) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL1817623 0.85 CYP3A4 (0.73) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL7504054 0.84 CYP3A4 (0.73) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL2193469 0.82 ATP4A (0.76) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL9746953 0.81 CYP3A4 (0.68) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL1813958 0.81 CYP3A4 (0.66) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971920-B1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-6265415-B1 ANTIULCER AGENT ASTRAZENECA AB (SE) 2001-07-24 US disclosed
EP-0971920-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION Astra Aktiebolag (SE) 2000-01-19 EP disclosed
WO-1998037080-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRA AKTIEBOLAG (SE) 1998-08-27 WO disclosed