SCHEMBL7499766

SCHEMBL7499766

COc1ccc2nc(OCc3ccccc3)nc(OCc3ccccc3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
EGFR P00533 2/20 0.51
ERBB2 P04626 1/20 0.51
MAOB P27338 2/20 0.50
TLR8 Q9NR97 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
NFKB1 P19838 1/20 0.47
RAB9A P51151 1/20 0.47
NFKB2 Q00653 1/20 0.47
KMT2A Q03164 1/20 0.47
RELA Q04206 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6471210 0.85 EGFR (0.50) ALDH1A1EGFRERBB2MAOBL3MBTL1
SCHEMBL7138839 0.81 EGFR (0.43) ALDH1A1EGFRERBB2MAOBL3MBTL1
SCHEMBL4725521 0.79 MAOB (0.48) ALDH1A1HTTEGFRERBB2MAOB
SCHEMBL30891765 0.78 NQO2 (0.46) ALDH1A1LMNAHTTNPSR1L3MBTL1
SCHEMBL2155868 0.77 ALDH1A1 (0.50) ALDH1A1LMNAHTTNPSR1EGFR
SCHEMBL15491330 0.76 EGFR (0.49) ALDH1A1EGFRERBB2MAOBL3MBTL1
Hydrochloric Acid SCHEMBL7123000 0.75 ALDH1A1 (0.51) ALDH1A1LMNAHTTNPSR1EGFR
SCHEMBL2420540 0.75 MAOB (0.44) ALDH1A1LMNAHTTNPSR1MAOB
SCHEMBL12324552 0.75 CNR2 (0.41) ALDH1A1LMNAHTTNPSR1MAOB
SCHEMBL28168224 0.75 MAOB (0.53) ALDH1A1NPSR1EGFRERBB2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607439-B1 NITROGENOUS HETEROCYCLIC COMPOUND EISAI CO LTD (JP) 2002-01-09 EP disclosed
US-6046206-A Method of treating a patient having a precancerous lesions with amide quinazoline derivatives CELL PATHWAYS, INC. (US) 2000-04-04 US disclosed
US-5801180-A ANTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS EISAI CO., LTD. (JP) 1998-09-01 US disclosed
US-5693652-A Benzimidazoles for ischemic heart conditions EISAI CO., LTD. (JP) 1997-12-02 US disclosed
US-5576322-A Anti-ischemic 2,4-diaminoquinazolines EISAI CO., LTD. (JP) 1996-11-19 US disclosed
EP-0607439-A1 NITROGENOUS HETEROCYCLIC COMPOUND Eisai Co., Ltd. (JP) 1994-07-27 EP disclosed