SCHEMBL7500428

SCHEMBL7500428

CC(C)(C)c1ccc2c(c1)C1(CCCNC1)C(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.49
PGR P06401 12/20 0.40
PDE4A P27815 4/20 0.38
PDE4B Q07343 4/20 0.38
PDE4C Q08493 4/20 0.38
PDE4D Q08499 4/20 0.38
PDE3B Q13370 4/20 0.38
PDE3A Q14432 4/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499439 0.90 BACE1 (0.47) BACE1PGRPDE4APDE4BPDE4C
SCHEMBL7504206 0.90 BACE1 (0.47) BACE1PGRPDE4APDE4BPDE4C
SCHEMBL7493171 0.90 BACE1 (0.47) BACE1PGRPDE4APDE4BPDE4C
SCHEMBL7501462 0.90 BACE1 (0.49) BACE1HTR2A
Hydrochloric Acid SCHEMBL7497244 0.89 BACE1 (0.46) BACE1PGRPDE4APDE4BPDE4C
SCHEMBL12056346 0.83 PGR (0.49) PGRPDE4APDE4BPDE4CPDE4D
SCHEMBL6637532 0.80 BACE1 (0.52) BACE1PGRPDE4APDE4BPDE4C
SCHEMBL6637484 0.80 PGR (0.54) BACE1PGRPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL6639312 0.78 BACE1 (0.51) BACE1PGRPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL6639499 0.78 PGR (0.53) BACE1PGRPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202994-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-05-08 EP claimed
WO-2001005790-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2001-01-25 WO claimed
EP-1202994-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-05-08 EP disclosed
WO-2001005790-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2001-01-25 WO disclosed