SCHEMBL7500755

SCHEMBL7500755

Cc1nc2c(N)cc(Cl)cn2c1C

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.35
PIK3R1 P27986 1/20 0.35
MAP3K14 Q99558 1/20 0.35
CYP3A4 P08684 13/20 0.34
CYP2C9 P11712 12/20 0.32
ALDH1A1 P00352 3/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32
CYP2C19 P33261 5/20 0.32
CYP2D6 P10635 5/20 0.32
CYP1A2 P05177 4/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6352105 0.81 CYP3A4 (0.33) MAP3K14CYP3A4CYP2C9ALDH1A1MAPT
SCHEMBL27824101 0.79 ALDH1A1 (0.31) CYP3A4CYP2C9ALDH1A1CYP2C19CYP2D6
SCHEMBL7498143 0.79 CYP3A4 (0.34) CYP3A4CYP2C9MEN1KMT2AMAPT
SCHEMBL4575125 0.79 APP (0.34) CYP3A4CYP2C9ALDH1A1MAPTCYP2C19
SCHEMBL6634450 0.76 ALDH1A1 (0.35) CYP3A4CYP2C9ALDH1A1MEN1KMT2A
SCHEMBL10396982 0.76 PIK3CD (0.33) PIK3CDPIK3R1MAP3K14
SCHEMBL4163641 0.73 CYP3A4 (0.49) CYP3A4CYP2C9ALDH1A1KMT2AMAPT
SCHEMBL6849960 0.73 CYP11B1 (0.32) CYP3A4CYP2C9ALDH1A1MAPTCYP2C19
Bromide SCHEMBL7554050 0.72 CYP3A4 (0.48) CYP3A4CYP2C9ALDH1A1KMT2AMAPT
SCHEMBL4888078 0.69 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971920-B1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-6265415-B1 ANTIULCER AGENT ASTRAZENECA AB (SE) 2001-07-24 US disclosed
EP-0971920-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION Astra Aktiebolag (SE) 2000-01-19 EP disclosed
WO-1998037080-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRA AKTIEBOLAG (SE) 1998-08-27 WO disclosed