SCHEMBL7500762

SCHEMBL7500762

CCOc1ccc(-c2cc(-c3cc(OC)c(OC)c(OC)c3)nc(N)c2C#N)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3A Q14432 2/20 0.69
KDM4E B2RXH2 8/20 0.65
NPSR1 Q6W5P4 4/20 0.65
HPGD P15428 3/20 0.65
MAPT P10636 4/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
ALDH1A1 P00352 3/20 0.58
ALOX15 P16050 2/20 0.58
MAPK1 P28482 1/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
HSD17B10 Q99714 1/20 0.58
GLA P06280 2/20 0.57
GAA P10253 1/20 0.57
GFER P55789 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
ADORA2A P29274 5/20 0.57
ADORA1 P30542 5/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7504723 0.92 PDE3A (0.58) PDE3AKDM4ENPSR1HPGDMAPT
SCHEMBL7501358 0.90 MEN1 (0.70) PDE3AKDM4ENPSR1HPGDMAPT
SCHEMBL7504766 0.87 KDM4E (0.60) PDE3AKDM4ENPSR1HPGDMAPT
SCHEMBL7507299 0.85 KDM4E (0.57) PDE3AKDM4ENPSR1HPGDMAPT
SCHEMBL7495415 0.84 KDM4E (0.56) PDE3AKDM4ENPSR1HPGDMAPT
SCHEMBL7507998 0.83 KDM4E (0.61) KDM4ENPSR1HPGDMAPTSMN1; SMN2
SCHEMBL7504091 0.82 KDM4E (0.60) KDM4ENPSR1HPGDMAPTSMN1; SMN2
SCHEMBL7509597 0.82 KDM4E (0.63) KDM4ENPSR1HPGDMAPTSMN1; SMN2
SCHEMBL7504138 0.82 KDM4E (0.60) KDM4ENPSR1HPGDMAPTMEN1
SCHEMBL7498392 0.80 PIM1 (0.76) PDE3AKDM4ENPSR1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222170-A1 NOVEL NICOTINONITRILE COMPOUNDS AstraZeneca AB (SE) 2002-07-17 EP claimed
WO-2001025207-A1 NOVEL NICOTINONITRILE COMPOUNDS ASTRAZENECA AB (SE) 2001-04-12 WO claimed