SCHEMBL7501358

SCHEMBL7501358

COc1ccc(-c2cc(-c3cc(OC)c(OC)c(OC)c3)nc(N)c2C#N)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.70
KMT2A Q03164 3/20 0.70
KDM4E B2RXH2 7/20 0.63
ALDH1A1 P00352 3/20 0.63
GLA P06280 2/20 0.63
MAPT P10636 2/20 0.63
GAA P10253 1/20 0.63
GFER P55789 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.63
ADORA2A P29274 8/20 0.62
ADORA1 P30542 8/20 0.62
NPSR1 Q6W5P4 4/20 0.62
HPGD P15428 2/20 0.62
RXFP1 Q9HBX9 2/20 0.61
TDP1 Q9NUW8 1/20 0.57
HSP90AA1 P07900 1/20 0.57
HSP90AB1 P08238 1/20 0.57
NPC1 O15118 1/20 0.54
BLM P54132 1/20 0.54
PDE3A Q14432 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507299 0.90 KDM4E (0.57) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7500762 0.90 PDE3A (0.69) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7553240 0.89 KDM4E (0.76) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL6250197 0.88 MEN1 (0.87) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7507998 0.88 KDM4E (0.61) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7504723 0.88 PDE3A (0.58) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7504091 0.87 KDM4E (0.60) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7504766 0.87 KDM4E (0.60) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7504138 0.87 KDM4E (0.60) MEN1KMT2AKDM4EALDH1A1GLA
SCHEMBL7509597 0.87 KDM4E (0.63) MEN1KMT2AKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222170-A1 NOVEL NICOTINONITRILE COMPOUNDS AstraZeneca AB (SE) 2002-07-17 EP claimed
WO-2001025207-A1 NOVEL NICOTINONITRILE COMPOUNDS ASTRAZENECA AB (SE) 2001-04-12 WO claimed
EP-1222188-A1 NOVEL IMIDAZOPYRIDINE CARBONITRILE COMPOUNDS AstraZeneca AB (SE) 2002-07-17 EP disclosed
WO-2001025237-A1 NOVEL IMIDAZOPYRIDINE CARBONITRILE COMPOUNDS ASTRAZENECA AB (SE) 2001-04-12 WO disclosed