SCHEMBL7501276

SCHEMBL7501276

CC(C)(C)OC(=O)Nc1ccc(OCCI)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.47
CYP2D6 P10635 1/20 0.44
MAPK14 Q16539 7/20 0.40
METAP1 P53582 1/20 0.38
AKT1 P31749 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MAPK12 P53778 4/20 0.38
TNF P01375 2/20 0.38
HCK P08631 1/20 0.38
MAPK13 O15264 2/20 0.38
MAPK11 Q15759 2/20 0.38
CDC25B P30305 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593957 0.88 AAK1 (0.47) AAK1CYP2D6MAPK14MAPK12TNF
SCHEMBL592972 0.88 AAK1 (0.47) AAK1CYP2D6MAPK14MAPK12TNF
SCHEMBL4689617 0.83 AAK1 (0.44) AAK1CYP2D6LMNAPOLBCDC25B
SCHEMBL6279532 0.82 BRD4 (0.48) AAK1CYP2D6
SCHEMBL593474 0.82 AAK1 (0.47) AAK1CYP2D6CDC25BMAPTSMN1; SMN2
SCHEMBL4252948 0.81 MAPK14 (0.52) MAPK14MAPK12TNFHCKMAPK13
SCHEMBL18593710 0.80 AAK1 (0.43) AAK1CYP2D6MAPK14LMNAPOLB
SCHEMBL4421726 0.80 CASP3 (0.47) AAK1CYP2D6LMNACDC25BMAPT
SCHEMBL6636004 0.79 AAK1 (0.42) AAK1CYP2D6LMNAPOLBCDC25B
SCHEMBL5257397 0.79 MAPK14 (0.65) MAPK14MAPK12TNFHCKMAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1232150-A1 UREA DERIVATIVES AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2002-08-21 EP disclosed
WO-2001036403-A1 UREA DERIVATIVES AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-05-25 WO disclosed