SCHEMBL7501713

SCHEMBL7501713

O=C(C=Cc1ncc[nH]1)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 2/20 0.50
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
MAPT P10636 5/20 0.46
MAOB P27338 3/20 0.45
MAOA P21397 2/20 0.44
RAB9A P51151 3/20 0.44
RECQL P46063 2/20 0.44
LMNA P02545 1/20 0.44
PTPN1 P18031 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
NPC1 O15118 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
TLR9 Q9NR96 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501707 1.00 CYP1B1 (0.50) CYP1B1ESR1ESR2MAPTMAOB
SCHEMBL7500978 0.86 F3 (0.53) CYP1B1ESR1ESR2MAPTMAOB
SCHEMBL7501752 0.86 KDM4E (0.51) CYP1B1MAPTMAOBMAOARAB9A
SCHEMBL7500993 0.86 F3 (0.53) CYP1B1ESR1ESR2MAPTMAOB
SCHEMBL7501747 0.86 KDM4E (0.51) CYP1B1MAPTMAOBMAOARAB9A
SCHEMBL7503829 0.85 CYP1B1 (0.50) CYP1B1MAPTMAOBMAOARAB9A
SCHEMBL7503643 0.85 SMN1; SMN2 (0.56) CYP1B1MAPTMAOBMAOALMNA
SCHEMBL3041754 0.85 CXCL12 (0.40) MAPTRAB9AALDH1A1NPC1MAPK1
SCHEMBL7503648 0.85 SMN1; SMN2 (0.56) CYP1B1MAPTMAOBMAOALMNA
SCHEMBL3041751 0.85 CXCL12 (0.40) MAPTRAB9AALDH1A1NPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0924202-B1 Imidazole derivative and medicine comprising the same as active ingredient SSP CO LTD (JP) 2002-05-29 EP disclosed
US-6071943-A IMMUNOMODULATORS WHICH SUPPRESS SPECIFIC CYTOKINES, FOR AUTOIMMUNE DISEASES SSP CO. LTD. (JP) 2000-06-06 US disclosed
EP-0924202-A1 Imidazole derivative and medicine comprising the same as active ingredient SSP Co., Ltd. (JP) 1999-06-23 EP disclosed