SCHEMBL7501957

SCHEMBL7501957

NS(=O)(=O)c1ccc(-c2oc(C(Cc3ccccc3)C(=O)O)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.54
PTGS1 P23219 4/20 0.54
CA2 P00918 4/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
NR4A2 P43354 2/20 0.41
CA1 P00915 2/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
CCR6 P51684 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5089153 0.90 PTGS2 (0.55) PTGS2PTGS1PTGDR2NR4A2
SCHEMBL7504823 0.89 PTGS2 (0.53) PTGS2PTGS1CA2PTGDR2CA1
SCHEMBL6002048 0.82 PTGS2 (0.50) PTGS2PTGS1CA2MAOAMAOB
SCHEMBL6002489 0.82 PTGS2 (0.50) PTGS2PTGS1CA2MAOAMAOB
SCHEMBL7504997 0.81 PTGS2 (0.63) PTGS2PTGS1CA2PTGDR2MAOA
SCHEMBL7499074 0.81 PTGS2 (0.62) PTGS2PTGS1CA2PTGDR2MAOA
SCHEMBL216120 0.80 PTGS2 (0.53) PTGS2PTGS1PTGDR2
SCHEMBL7501237 0.78 PTGS2 (0.61) PTGS2PTGS1CA2MAOAMAOB
SCHEMBL7505500 0.78 PTGS2 (0.61) PTGS2PTGS1CA2MAOAMAOB
SCHEMBL9029716 0.77 PTGS2 (0.59) PTGS2PTGS1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699192-B1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-07-24 EP claimed