SCHEMBL7511036

SCHEMBL7511036

C[Si](C)(C)CCOCn1nc(/C=C/c2ccccc2)c2cc(/C=C/c3ccccc3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.36
IP6K1 Q92551 3/20 0.34
EGFR P00533 1/20 0.33
IP6K3 Q96PC2 1/20 0.33
IP6K2 Q9UHH9 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
ENPP2 Q13822 1/20 0.31
TUBB1 Q9H4B7 1/20 0.31
KDR P35968 1/20 0.31
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
RAB9A P51151 3/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
RELA Q04206 2/20 0.31
PKM P14618 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
GAA P10253 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5512063 1.00 NPC1 (0.36) NPC1IP6K1EGFRIP6K3IP6K2
SCHEMBL14493368 0.91 CHEK1 (0.39) NPC1EGFRKDRCHEK1
SCHEMBL14493340 0.91 SMN1; SMN2 (0.37) NPC1EGFRCYP1A2TUBB1KDR
SCHEMBL5526396 0.91 CHEK1 (0.39) NPC1EGFRKDRCHEK1
SCHEMBL14493369 0.90 ENPP2 (0.37) NPC1EGFRENPP2TUBB1KDM4E
SCHEMBL14493379 0.90 NPC1 (0.35) NPC1EGFRTUBB1
SCHEMBL27615251 0.90 CNR1 (0.37) NPC1EGFRKDRKDM4EALDH1A1
SCHEMBL5523225 0.90 ENPP2 (0.37) NPC1EGFRENPP2TUBB1KDM4E
SCHEMBL3707196 0.85 ENPP2 (0.37) NPC1IP6K1EGFRCYP1A2ENPP2
SCHEMBL3707199 0.85 ENPP2 (0.37) NPC1IP6K1EGFRCYP1A2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7232912-B2 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation AGOURON PHARMACEUTICALS, INC. (US) 2007-06-19 US disclosed
US-7232912-B2 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation AGOURON PHARMACEUTICALS, INC. (US) 2007-06-19 US disclosed
EP-1250326-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2002-10-23 EP disclosed
WO-2001053268-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed