SCHEMBL7511468

SCHEMBL7511468

CC(NOC(N)=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.49
HDAC4 P56524 3/20 0.49
HDAC1 Q13547 3/20 0.49
HDAC6 Q9UBN7 3/20 0.47
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
APAF1 O14727 1/20 0.46
KMT2A Q03164 3/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 2/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALOX5 P09917 1/20 0.44
PARP1 P09874 1/20 0.44
HPGD P15428 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28010037 0.83 HDAC6 (0.49) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL27821681 0.83 HDAC6 (0.49) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL27882319 0.81 HDAC6 (0.47) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL27845616 0.80 HDAC6 (0.46) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL26461278 0.80 TSHR (0.52) ALDH1A1HSD17B10APAF1KMT2ALMNA
SCHEMBL18922945 0.77 HDAC6 (0.44) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL28493114 0.76 KMT2A (0.47) HDAC3HDAC4HDAC1ALDH1A1HSD17B10
SCHEMBL28493115 0.76 KMT2A (0.47) HDAC3HDAC4HDAC1ALDH1A1HSD17B10
SCHEMBL9209754 0.76 MEN1 (0.47) HSD17B10APAF1KMT2AMEN1PKM
SCHEMBL28712237 0.76 KMT2A (0.43) HDAC3HDAC4HDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951284-A4 PHENYLETHYLAMINE DERIVATIVES TEVA PHARMA (IL) 2002-03-20 EP disclosed
EP-0951284-A1 PHENYLETHYLAMINE DERIVATIVES TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 1999-10-27 EP disclosed
WO-1998026775-A1 PHENYLETHYLAMINE DERIVATIVES TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 1998-06-25 WO disclosed