SCHEMBL7512290

SCHEMBL7512290

O=C(C1CCCN1Cc1ccccc1)N1CCN(Cc2ccc(F)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
FAAH O00519 1/20 0.54
MCHR1 Q99705 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TSHR P16473 1/20 0.52
SIGMAR1 Q99720 2/20 0.52
ATM Q13315 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678657 1.00 KDM4E (0.55) KDM4EFAAHMCHR1MEN1KMT2A
Hydrochloric Acid SCHEMBL7517966 0.86 MCHR1 (0.68) KDM4EMCHR1
Hydrochloric Acid SCHEMBL6680315 0.86 MCHR1 (0.68) KDM4EMCHR1
Hydrochloric Acid SCHEMBL6658225 0.85 MEN1 (0.53) KDM4EMCHR1MEN1KMT2A
Hydrochloric Acid SCHEMBL6662216 0.85 MEN1 (0.53) KDM4EMCHR1MEN1KMT2A
Hydrochloric Acid SCHEMBL6662222 0.85 MEN1 (0.53) KDM4EMCHR1MEN1KMT2A
SCHEMBL6908168 0.84 L3MBTL1 (0.50)
SCHEMBL6659429 0.84 L3MBTL1 (0.50)
SCHEMBL1190538 0.84 MCHR1 (0.63) KDM4EMCHR1MEN1KMT2ATSHR
SCHEMBL7473424 0.84 MCHR1 (0.63) KDM4EMCHR1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257544-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE Vertex Pharmaceuticals Incorporated (US) 2002-11-20 EP disclosed
WO-2001058891-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-08-16 WO disclosed