SCHEMBL7512508

SCHEMBL7512508

N[C@H](Cc1ccccc1)C(=O)NC(=O)[C@@H]1CCCN1Cc1ncccc1-n1cncn1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F2 P00734 6/20 0.50
TPH1 P17752 1/20 0.42
ACE P12821 1/20 0.38
NAMPT P43490 2/20 0.38
HSD11B1 P28845 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
DPP4 P27487 2/20 0.35
DPP8 Q6V1X1 2/20 0.35
DPP9 Q86TI2 2/20 0.35
DPP7 Q9UHL4 2/20 0.35
FAP Q12884 1/20 0.35
MC3R P41968 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
CCR4 P51679 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6077661 0.99 F2 (0.49) F2TPH1ACENAMPTHSD11B1
Hydrochloric Acid SCHEMBL6079169 0.89 F2 (0.59) F2TPH1ACENPSR1DPP4
SCHEMBL6078139 0.83 F2 (0.61) F2TPH1MC3R
SCHEMBL7512500 0.80 F2 (0.61) F2DPP4DPP8DPP9DPP7
Hydrochloric Acid SCHEMBL6077658 0.79 F2 (0.60) F2ACEDPP4DPP8DPP9
SCHEMBL6078129 0.76 F2 (0.60) F2TPH1ACENPSR1
SCHEMBL7513994 0.76 F2 (0.60) F2TPH1ACENPSR1
Hydrochloric Acid SCHEMBL6077070 0.75 F2 (0.59) F2TPH1ACENPSR1
SCHEMBL7102501 0.75 F2 (0.49) F2ACENPSR1DPP4DPP8
SCHEMBL7107001 0.75 CCR4 (0.49) F2ACENPSR1DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002064559-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed