SCHEMBL751258

SCHEMBL751258

C[Si](C)(C)C#Cc1ccc(-c2cnc(C3CC(F)(F)CN3C(=O)O)[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PRCP P42785 11/20 0.42
CYP3A4 P08684 3/20 0.37
CYP2C9 P11712 3/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 1/20 0.35
HCRTR1 O43613 3/20 0.34
HCRTR2 O43614 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2706903 0.87 PRCP (0.43) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL203457 0.87 PRCP (0.43) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL204580 0.83 CYP3A4 (0.59) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2707746 0.83 CYP3A4 (0.59) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL750686 0.81 CYP3A4 (0.40) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL12295933 0.80 PRCP (0.45) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL28059665 0.79 PRCP (0.46) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL1478863 0.76 CYP3A4 (0.39) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL541070 0.76 CYP3A4 (0.39) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL1478321 0.76 PRCP (0.37) PRCPCYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed