SCHEMBL28059665

SCHEMBL28059665

C[Si](C)(C)CC(=O)Cc1ccc(-c2cnc(C3CC(F)(F)CN3C(=O)O)[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRCP P42785 11/20 0.46
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP1A2 P05177 1/20 0.38
NR1I2 O75469 1/20 0.36
ABCB11 O95342 1/20 0.36
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL751258 0.79 PRCP (0.42) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL9980237 0.73 PRCP (0.45) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL883052 0.73 PRCP (0.48) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL19578300 0.72 PRCP (0.46) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL12175097 0.70 KCNH2 (0.50) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL12175082 0.70 KCNH2 (0.62) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL12175205 0.70 CYP3A4 (0.58) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL2708425 0.70 PRCP (0.51) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL205053 0.70 PRCP (0.51) PRCPCYP3A4CYP2C9CYP1A2NR1I2
SCHEMBL752316 0.70 MAPK13 (0.41) PRCPCYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104016971-B Antiviral compound PHARMASSET INC. (US) 2016-05-25 CN disclosed