SCHEMBL7513604

SCHEMBL7513604

O=C(Nc1ccc(C(F)(F)F)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.83
PTGS1 P23219 3/20 0.83
NPC1 O15118 2/20 0.82
RAB9A P51151 2/20 0.82
RORC P51449 1/20 0.80
EPHX2 P34913 2/20 0.70
HDAC3 O15379 1/20 0.70
HDAC8 Q9BY41 1/20 0.70
HDAC6 Q9UBN7 1/20 0.70
TRPV4 Q9HBA0 1/20 0.67
MAPT P10636 2/20 0.66
XBP1 P17861 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
KCNQ3 O43525 1/20 0.66
KCNQ2 O43526 1/20 0.66
KCNE1 P15382 1/20 0.66
KCNQ1 P51787 1/20 0.66
MEN1 O00255 1/20 0.65
LMNA P02545 1/20 0.65
KMT2A Q03164 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2064051 0.93 TRPV1 (0.73) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL2923145 0.93 TRPV1 (0.73) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL674439 0.93 HDAC6 (0.82) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL11730950 0.93 NPC1 (0.77) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL15948139 0.91 TRPV1 (0.76) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL96039 0.91 TRPV1 (0.71) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL28910371 0.91 TRPV1 (0.71) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL95224 0.91 TRPV1 (0.71) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL22721382 0.91 PTGS1 (0.76) TRPV1PTGS1NPC1RAB9ARORC
SCHEMBL7557294 0.91 TRPV1 (1.00) TRPV1PTGS1NPC1RAB9ARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001021160-B1 CARBOXYMIDE AND ANILINE DERIVATIVES AS SELECTIVE INHIBITORS OF PATHOGENS AXXIMA PHARMACEUTICALS AG (DE) 2002-05-30 WO claimed