SCHEMBL7513684

SCHEMBL7513684

CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCNC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.51
CTSS P25774 3/20 0.51
CTSL P07711 2/20 0.51
CTSB P07858 1/20 0.51
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CAPN1 P07384 1/20 0.46
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
AAK1 Q2M2I8 1/20 0.42
MAPK1 P28482 1/20 0.41
REN P00797 2/20 0.40
MAP1LC3B Q9GZQ8 1/20 0.40
MAP1LC3A Q9H492 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PSMB5 P28074 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8133234 0.86 HDAC4 (0.52) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL8133237 0.86 HDAC4 (0.52) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL6582894 0.85 CTSK (0.48) CTSKCTSSCTSLCTSBHDAC4
SCHEMBL8121033 0.84 KMT2A (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL8387090 0.84 KMT2A (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL8121031 0.84 KMT2A (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL4320742 0.83 CTSK (0.46) CTSKCTSSCTSLCTSBHDAC4
SCHEMBL4320739 0.83 CTSK (0.46) CTSKCTSSCTSLCTSBHDAC4
SCHEMBL4310648 0.82 CTSK (0.47) CTSKCTSSCTSLCTSBHDAC4
SCHEMBL5099466 0.82 CTSK (0.47) CTSKCTSSCTSLCTSBHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991753-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2001-07-11 EP disclosed
EP-0991753-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-04-12 EP disclosed
WO-1998050534-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-12 WO disclosed