SCHEMBL7513830

SCHEMBL7513830

CC(=O)O[C@H]1CC[C@H](Nc2nc(N)ncc2Sc2ccc(Cl)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.49
NPY5R Q15761 2/20 0.41
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
MAPK3 P27361 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SYK P43405 3/20 0.36
CHEK1 O14757 2/20 0.35
MAPKAPK2 P49137 2/20 0.35
CSNK2A1 P68400 1/20 0.35
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
MAPK8 P45983 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7524053 0.90 RXFP1 (0.47) RXFP1NPY5RHTR1ADRD2DRD4
SCHEMBL7521012 0.90 RXFP1 (0.47) RXFP1HTR1ADRD2DRD4MAPK3
SCHEMBL7514853 0.89 RXFP1 (0.46) RXFP1NPY5RHTR1ADRD2DRD4
SCHEMBL7514857 0.89 RXFP1 (0.46) RXFP1NPY5RHTR1ADRD2DRD4
SCHEMBL7520253 0.87 RXFP1 (0.44) RXFP1HTR1ADRD2DRD4MAPK3
SCHEMBL7510904 0.83 RXFP1 (0.51) RXFP1HTR1ADRD2DRD4SYK
SCHEMBL7510908 0.83 RXFP1 (0.51) RXFP1HTR1ADRD2DRD4SYK
SCHEMBL7515467 0.81 RXFP1 (0.48) RXFP1HTR1ADRD2DRD4SYK
SCHEMBL7515471 0.81 RXFP1 (0.48) RXFP1HTR1ADRD2DRD4SYK
SCHEMBL7513904 0.79 RXFP1 (0.49) RXFP1HTR1ADRD2DRD4SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP claimed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO claimed
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed