SCHEMBL7515253

SCHEMBL7515253

CC(c1cc([N+](=O)[O-])ccc1Oc1ccc(Cl)c(Cl)c1)N(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.47
SLC6A4 P31645 4/20 0.47
KCNH2 Q12809 4/20 0.47
ALDH1A1 P00352 4/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
GAA P10253 2/20 0.45
PKM P14618 1/20 0.45
PDE7A Q13946 1/20 0.43
HSD17B10 Q99714 1/20 0.42
TBXA2R P21731 1/20 0.41
MAPT P10636 4/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.40
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
KDM4E B2RXH2 2/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152328 0.87 HTR2A (0.43) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL7515248 0.79 TBXA2R (0.47) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL6151967 0.79 HTR2A (0.66) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL7454203 0.78 HTR2A (0.50) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL6151964 0.78 PDE7A (0.49) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL6151811 0.75 MEN1 (0.55) ALDH1A1MEN1KMT2AGAAPKM
SCHEMBL5836477 0.74 SLC6A4 (0.66) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL7457814 0.73 SLC6A4 (0.42) HTR2ASLC6A4KCNH2ALDH1A1MAPT
SCHEMBL13860469 0.73 HSD17B10 (0.54) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL22069594 0.71 HSPB1 (0.61) ALDH1A1MEN1KMT2AGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1220831-A1 BIARYL ETHER DERIVATIVES USEFUL AS MONOAMINE REUPTAKE INHIBITORS Pfizer Products Inc. (US) 2002-07-10 EP disclosed
WO-2001027068-A1 BIARYL ETHER DERIVATIVES USEFUL AS MONOAMINE REUPTAKE INHIBITORS PFIZER PRODUCTS INC. (US) 2001-04-19 WO disclosed