SCHEMBL7516614

SCHEMBL7516614

N#Cc1ccc(COC[C@@H](OCc2ccc(C#N)cc2)[C@@H](O)[C@H](O)[C@@H](COCc2ccc(C#N)cc2)OCc2ccc(C#N)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.42
MAOB P27338 2/20 0.39
LOXL2 Q9Y4K0 2/20 0.38
CYP2A6 P11509 1/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CA2 P00918 3/20 0.37
CA9 Q16790 2/20 0.37
CA12 O43570 1/20 0.37
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA14 Q9ULX7 1/20 0.37
GAA P10253 1/20 0.36
CHRM3 P20309 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
GBA1 P04062 1/20 0.35
UGCG Q16739 1/20 0.35
GBA2 Q9HCG7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452032 0.94 MAOB (0.49) ALOX5MAOBRAB9ANPC1SMN1; SMN2
SCHEMBL7510108 0.94 MAOB (0.49) ALOX5MAOBRAB9ANPC1SMN1; SMN2
SCHEMBL7450464 0.84 MAOB (0.41) ALOX5MAOBLOXL2CYP2A6RAB9A
SCHEMBL7989854 0.83 AR (0.39) MAOBRAB9ANPC1SMN1; SMN2L3MBTL1
SCHEMBL7510253 0.82 SMPD1 (0.49)
SCHEMBL7510889 0.79 KCNH2 (0.44) MAOBRAB9ANPC1SMN1; SMN2CA2
SCHEMBL7992780 0.79 IDO1 (0.41) ALOX5MAOBRAB9ASMN1; SMN2CA2
SCHEMBL5742123 0.78 CA1 (0.56) CA2CA9CA1CA7
SCHEMBL7968710 0.78 ALOX5 (0.44) ALOX5MAOBLOXL2CYP2A6RAB9A
SCHEMBL7968714 0.78 ALOX5 (0.44) ALOX5MAOBLOXL2CYP2A6RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175385-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Pharmacor Inc. (CA) 2002-01-30 EP disclosed
US-6313177-B1 AS ANTIVIRAL AGENTS PHARMACOR INC. (CA) 2001-11-06 US disclosed
WO-2001029014-A1 ISOTHIAZOLE-5-CARBOXYLIC ESTERS AS MICROBICIDES NIHON BAYER AGROCHEM K.K. (JP) 2001-04-26 WO disclosed
WO-2000066524-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PHARMACOR INC. (CA) 2000-11-09 WO disclosed