SCHEMBL7517952

SCHEMBL7517952

COC(=O)c1ccc([N+](=O)[O-])cc1OCCO[Si](C)(C)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.41
ADRB1 P08588 2/20 0.41
ADRB3 P13945 2/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP2C19 P33261 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 2/20 0.39
HTT P42858 2/20 0.39
PKM P14618 1/20 0.39
LMNA P02545 1/20 0.39
CYP19A1 P11511 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7525234 0.94 TSHR (0.41) ADRB2ADRB1ADRB3ALDH1A1CYP2C19
SCHEMBL30727333 0.83 TSHR (0.49) ALDH1A1TSHRTDP1KMT2AMEN1
SCHEMBL1185010 0.83 TSHR (0.49) ALDH1A1TSHRTDP1KMT2AMEN1
SCHEMBL223562 0.82 LMNA (0.51) ALDH1A1CYP2C19TDP1KMT2ANPC1
SCHEMBL7006661 0.82 MAPT (0.50) ALDH1A1CYP2C19TDP1KMT2ANPC1
SCHEMBL5103038 0.81 S1PR4 (0.41) ALDH1A1CYP2C19TSHRTDP1KMT2A
SCHEMBL7520954 0.81 TSHR (0.42) ALDH1A1CYP2C19TSHRTDP1KMT2A
SCHEMBL30326242 0.80 S1PR4 (0.40) ALDH1A1CYP2C19TSHRTDP1KMT2A
SCHEMBL12134869 0.80 CYP19A1 (0.42) ALDH1A1CYP2C19TSHRTDP1KMT2A
SCHEMBL2909665 0.80 MAPT (0.44) ALDH1A1CYP2C19TSHRTDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173414-A1 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2002-01-23 EP disclosed
WO-2000064864-A9 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RES CAMPAIGN TECH (GB) 2001-12-27 WO disclosed
WO-2000064864-A1 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-11-02 WO disclosed