SCHEMBL752049

SCHEMBL752049

C#Cc1ccc(-c2cnc(C3CC(F)(F)CN3C(=O)CC(C)CNC(=O)OC)[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRCP P42785 8/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2C9 P11712 4/20 0.41
KCNH2 Q12809 3/20 0.41
NR1I2 O75469 2/20 0.41
ABCB11 O95342 1/20 0.41
OPRK1 P41145 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 1/20 0.39
F11 P03951 3/20 0.33
F2 P00734 1/20 0.32
ACACB O00763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL752515 0.92 CYP3A4 (0.41) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL750686 0.90 CYP3A4 (0.40) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL751612 0.86 CYP3A4 (0.56) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL205384 0.82 CYP3A4 (0.61) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL2706896 0.82 CYP3A4 (0.61) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL751761 0.82 CYP3A4 (0.43) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL751733 0.82 CYP3A4 (0.62) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL19578300 0.79 PRCP (0.46) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL750283 0.76 PRCP (0.40) PRCPCYP3A4CYP2C9KCNH2NR1I2
SCHEMBL751564 0.76 PRCP (0.42) PRCPCYP3A4CYP2C9KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed