SCHEMBL7521622

SCHEMBL7521622

O=[N+]([O-])c1ccc(C(Br)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
LMNA P02545 1/20 0.58
KMT2A Q03164 4/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
MEN1 O00255 3/20 0.50
CRHBP P24387 1/20 0.50
ATM Q13315 1/20 0.50
CRHR2 Q13324 1/20 0.50
TLR9 Q9NR96 1/20 0.50
HPGD P15428 1/20 0.50
ALOX12 P18054 1/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
MAPK1 P28482 2/20 0.44
CYP1A2 P05177 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
POLB P06746 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9068786 0.92 ALDH1A1 (0.52) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL11795354 0.88 ALDH1A1 (0.58) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL5827237 0.86 ALDH1A1 (0.60) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL5663512 0.83 ALDH1A1 (0.62) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL3695529 0.83 ALDH1A1 (0.62) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL2601112 0.82 ALDH1A1 (0.60) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL19334711 0.82 ALDH1A1 (0.60) ALDH1A1LMNAKMT2AL3MBTL1MEN1
Nitrobenzene SCHEMBL9700705 0.81 ALDH1A1 (0.80) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL3258821 0.80 ALDH1A1 (0.58) ALDH1A1LMNAKMT2AL3MBTL1MEN1
SCHEMBL1813716 0.80 CA12 (0.58) ALDH1A1LMNAKMT2AL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417213-B2 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-09 US disclosed
US-20020006944-A1 Tricyclic compounds, their production and use OHKAWA SHIGENORI (JP) 2002-01-17 US disclosed
EP-1112251-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2001-07-04 EP disclosed
US-6248766-B1 CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-19 US disclosed
WO-2000015609-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA S.A. (FR) 2000-03-23 WO disclosed
EP-0929534-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS Takeda Pharmaceutical Company Limited (JP) 1999-07-21 EP disclosed
WO-1998013356-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020006944-A1 Tricyclic compounds, their production and use CNR1, PTGER1, PTGDR ALDH1A1 1662/4885LMNA 2418/4885KMT2A 3081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.