SCHEMBL7522342

SCHEMBL7522342

CC(C)C[C@H](NC(=O)Nc1cccc2ccccc12)C(=O)NC1CCOC1O

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 14/20 0.65
ANPEP P15144 1/20 0.64
CASP1 P29466 5/20 0.53
CASP3 P42574 4/20 0.51
CASP7 P55210 4/20 0.51
CASP6 P55212 3/20 0.51
CASP8 Q14790 3/20 0.51
CAPNS1 P04632 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520605 1.00 CAPN1 (0.65) CAPN1ANPEPCASP1CASP3CASP7
SCHEMBL7512325 0.88 ANPEP (0.60) CAPN1ANPEPCASP1CASP3CASP7
SCHEMBL7513408 0.86 ANPEP (0.58) CAPN1ANPEPCASP1CASP3CASP7
SCHEMBL8808063 0.85 CASP1 (0.72) CAPN1CASP1CASP3CASP7CASP6
SCHEMBL8808053 0.85 CASP1 (0.72) CAPN1CASP1CASP3CASP7CASP6
SCHEMBL8812444 0.84 CASP1 (0.73) CAPN1CASP1CASP3CASP7CASP6
SCHEMBL8812448 0.84 CASP1 (0.73) CAPN1CASP1CASP3CASP7CASP6
SCHEMBL6770677 0.82 CAPN1 (0.75) CAPN1CASP3CAPNS1
SCHEMBL7515616 0.81 ANPEP (0.64) ANPEPCASP1CASP3CASP7CASP6
SCHEMBL8807569 0.80 CAPN1 (0.55) CAPN1CASP1CASP3CASP7CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed
US-5496834-A PEPTIDE DERIVATIVES AS CATHEPSIN L INHIBITORS AND INHIBITORS OF BONE RESORPTION OR TREATMENT OF OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
EP-0641800-A1 Lactol derivatives as inhibiters of cathepsin L Takeda Chemical Industries, Ltd. (JP) 1995-03-08 EP disclosed