SCHEMBL7522654

SCHEMBL7522654

CCOP(=O)(OCC)C(=CC=Cc1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)P(=O)(OCC)OCC

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.71
NR1I2 O75469 2/20 0.71
GABBR2 O75899 2/20 0.52
GABBR1 Q9UBS5 2/20 0.52
PTGS1 P23219 4/20 0.43
PTGS2 P35354 4/20 0.43
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
GPR55 Q9Y2T6 1/20 0.39
ALOX5 P09917 2/20 0.38
HTT P42858 1/20 0.38
EEF2K O00418 1/20 0.38
SRC P12931 1/20 0.38
LMNA P02545 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL678403 0.83 HMGCR (1.00) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7139090 0.82 HMGCR (0.71) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7519377 0.80 GABBR2 (0.61) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL12160467 0.77 HMGCR (0.77) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7134494 0.76 HMGCR (0.85) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7137096 0.76 HMGCR (0.83) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7083282 0.76 HMGCR (0.83) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL9390686 0.73 HMGCR (0.50) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL7521931 0.73 HMGCR (0.80) HMGCRNR1I2GABBR2GABBR1PTGS1
SCHEMBL17407580 0.73 HMGCR (0.70) HMGCRNR1I2GABBR2GABBR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0845991-B1 USE OF PHENOL SUBSTITUTED DIPHOSPHONATES AS ANTINEOPLASTIC AGENTS SYMPHAR SA (CH) 2002-02-06 EP claimed
EP-0845991-A2 USE OF PHENOL SUBSTITUTED DIPHOSPHONATES AS ANTINEOPLASTIC AGENTS SYMPHAR S.A. (CH) 1998-06-10 EP claimed
WO-1997004785-A1 USE OF PHENOL SUBSTITUTED DIPHOSPHONATES AS ANTINEOPLASTIC AGENTS SYMPHAR S.A. (CH) 1997-02-13 WO claimed
US-5128331-A Gen-diphosphonates SYMPHAR S.A. (CH) 1992-07-07 US disclosed
US-5043330-A Antiinflammatory and hypotensive agents; antihyperlipemia SYMPHAR S.A. (CH) 1991-08-27 US disclosed