SCHEMBL7522772

SCHEMBL7522772

COc1ccc(CNc2nc(-c3cnccn3)nc3sc(C)cc23)cc1Cl.Cc1cc2c(Cl)nc(-c3cnccn3)nc2s1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCDIN3D Q7Z5W3 2/20 0.42
PDE5A O76074 13/20 0.42
NPC1 O15118 1/20 0.38
GALR3 O60755 1/20 0.38
NR2F2 P24468 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5117610 0.97 PDE5A (0.42) BCDIN3DPDE5ANPC1GALR3NR2F2
SCHEMBL7508291 0.92 BCDIN3D (0.42) BCDIN3DPDE5A
SCHEMBL5128040 0.89 PDE5A (0.43) BCDIN3DPDE5A
SCHEMBL5122834 0.89 NPC1 (0.48) PDE5ANPC1GALR3NR2F2RAB9A
SCHEMBL5114999 0.87 PRKCI (0.43) BCDIN3DPDE5A
SCHEMBL5128521 0.87 ADORA2A (0.49)
SCHEMBL7512073 0.87 MAPT (0.47) BCDIN3DPDE5A
SCHEMBL5113662 0.85 PDE5A (0.47) PDE5ANPC1
SCHEMBL5115283 0.85 PDE5A (0.45) BCDIN3DPDE5A
SCHEMBL7504877 0.84 MAPT (0.41) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920431-A1 THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 1999-06-09 EP disclosed
WO-1998006722-A1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed