SCHEMBL7523835

SCHEMBL7523835

Fc1nc2ccccc2c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 3/20 0.54
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 7/20 0.46
ALDH1A1 P00352 3/20 0.46
GLA P06280 3/20 0.46
MAOA P21397 2/20 0.46
HPGD P15428 2/20 0.46
CASP1 P29466 2/20 0.46
CASP7 P55210 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CHRM1 P11229 1/20 0.46
NQO2 P16083 1/20 0.46
DRD1 P21728 1/20 0.46
ACHE P22303 1/20 0.46
SLC6A2 P23975 1/20 0.46
ADRA1A P35348 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30528247 0.78 KDM4E (0.44) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL3237036 0.78 KDM4E (0.44) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL15058512 0.78 KDM4E (0.44) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL28360035 0.76 KDM4E (0.43) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL5096456 0.75 MAPT (0.62) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL4003840 0.75 DCPS (0.63) KMT2AKDM4EALDH1A1GLAMAOA
SCHEMBL29058640 0.75 KDM4E (0.42) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL11690509 0.74 KDM4E (0.56) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL538767 0.73 KDM4E (0.40) GPR3KMT2AKDM4EALDH1A1GLA
SCHEMBL15514447 0.73 KDM4E (0.40) GPR3KMT2AKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946513-B1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 2002-01-30 EP claimed
US-6120703-A Derivatives of 6-fluorophenanthridine for liquid crystal mixtures AVENTIS RESEARCH & TECHNOLOGIES DEUTSCHLAND GMBH & CO. KG (DE) 2000-09-19 US claimed
EP-0946513-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES Aventis Research & Technologies GmbH & Co. KG (DE) 1999-10-06 EP claimed
WO-1998027060-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO KG (DE) 1998-06-25 WO claimed
EP-0946513-B1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 2002-01-30 EP disclosed
EP-0946513-B1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 2002-01-30 EP disclosed
US-6120703-A Derivatives of 6-fluorophenanthridine for liquid crystal mixtures AVENTIS RESEARCH & TECHNOLOGIES DEUTSCHLAND GMBH & CO. KG (DE) 2000-09-19 US disclosed
US-6120703-A Derivatives of 6-fluorophenanthridine for liquid crystal mixtures AVENTIS RESEARCH & TECHNOLOGIES DEUTSCHLAND GMBH & CO. KG (DE) 2000-09-19 US disclosed
US-6120703-A Derivatives of 6-fluorophenanthridine for liquid crystal mixtures AVENTIS RESEARCH & TECHNOLOGIES DEUTSCHLAND GMBH & CO. KG (DE) 2000-09-19 US disclosed
EP-0946513-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES Aventis Research & Technologies GmbH & Co. KG (DE) 1999-10-06 EP disclosed
EP-0946513-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES Aventis Research & Technologies GmbH & Co. KG (DE) 1999-10-06 EP disclosed
EP-0799207-B1 PROCESS FOR THE PREPARATION OF FLUORINATED HETEROCYCLIC COMPOUNDS F2 CHEMICALS LIMITED (GB) 1999-06-09 EP disclosed
US-5859255-A Process for the preparation of fluorinated heterocyclic compounds F2 CHEMICALS LTD. (GB) 1999-01-12 US disclosed
WO-1998027060-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO KG (DE) 1998-06-25 WO disclosed
WO-1998027060-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO KG (DE) 1998-06-25 WO disclosed
CN-1170406-A Preparation of fluorinated heterocyclic compounds F2 CHEMICAL PRODUCTS LTD (GB) 1998-01-14 CN disclosed
EP-0799207-A1 PROCESS FOR THE PREPARATION OF FLUORINATED HETEROCYCLIC COMPOUNDS BNFL FLUOROCHEMICALS LTD. (GB) 1997-10-08 EP disclosed
WO-1996019456-A1 PROCESS FOR THE PREPARATION OF FLUORINATED HETEROCYCLIC COMPOUNDS BNFL FLUOROCHEMICALS LTD. (GB) 1996-06-27 WO disclosed