SCHEMBL752460

SCHEMBL752460

CCOC(=O)Cc1ccno1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.43
TRPM8 Q7Z2W7 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NPC1 O15118 1/20 0.40
PKM P14618 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
LMNA P02545 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27908114 0.84 CYP1A2 (0.47) SMN1; SMN2HSD17B10L3MBTL1CYP3A4CYP2C9
SCHEMBL2822798 0.82 CYP4F2 (0.41) SMN1; SMN2HSD17B10NPC1PKMNFKB1
SCHEMBL27503059 0.74 KMT2A (0.47) SMN1; SMN2HSD17B10NPC1RAB9AL3MBTL1
SCHEMBL1650609 0.74
SCHEMBL1415222 0.73 GAA (0.44) SMN1; SMN2PKMCYP3A4CYP2C9ALDH1A1
SCHEMBL4751904 0.72 VHL (0.54) SMN1; SMN2PKMRAB9AALDH1A1CA12
SCHEMBL25601889 0.72 KLK7 (0.41) SMN1; SMN2TRPM8ALDH1A1CA12CA1
SCHEMBL11102141 0.72
SCHEMBL14205589 0.71 ALDH1A1 (0.51) HSD17B10CYP3A4CYP2C9ALDH1A1LMNA
SCHEMBL916156 0.71 HDAC4 (0.50) SMN1; SMN2PKMCYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430012-A1 7-AZA-SPIRO[3.5]NONANE-7-CARBOXYLATE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-21 EP disclosed
WO-2010130945-A1 7-AZA-SPIRO[3.5]NONANE-7-CARBOXYLATE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-11-18 WO disclosed