SCHEMBL7525302

SCHEMBL7525302

COc1ccc2c(ccc3ccc4c(c32)C(c2ccc(OCCN3CCCCC3)cc2)c2ccccc2-4)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 12/20 0.71
ESR2 Q92731 10/20 0.71
HRH3 Q9Y5N1 5/20 0.49
EBP Q15125 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
PGR P06401 1/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44
DRD1 P21728 1/20 0.44
TBXA2R P21731 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966174 0.94 ESR1 (0.80) ESR1ESR2HRH3PGRCHRM2
SCHEMBL7524349 0.90 ESR1 (0.88) ESR1ESR2HRH3
SCHEMBL8610437 0.89 ESR1 (0.86) ESR1ESR2HRH3
SCHEMBL8966218 0.87 ESR1 (0.76) ESR1ESR2HRH3
SCHEMBL7525280 0.86 ESR1 (0.69) ESR1ESR2
SCHEMBL7528598 0.85 ESR1 (0.67) ESR1ESR2HRH3PGRCHRM2
SCHEMBL8966242 0.84 ESR1 (0.68) ESR1ESR2HRH3EBPSIGMAR1
SCHEMBL8965793 0.84 ESR1 (0.68) ESR1ESR2HRH3EBPSIGMAR1
SCHEMBL8966205 0.83 ESR1 (1.00) ESR1ESR2HRH3
SCHEMBL7527242 0.83 ESR1 (0.66) ESR1ESR2HRH3EBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832882-B1 Naphthofluorene compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2002-04-03 EP disclosed
EP-0832882-A2 Naphthofluorene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed