SCHEMBL7526237

SCHEMBL7526237

NC(=O)c1cccc(CCCN2CCOCC2)c1C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.54
PARP2 Q9UGN5 2/20 0.54
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTR7 P34969 2/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
ABCB1 P08183 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7527733 0.92 PARP1 (0.53) PARP1PARP2ALDH1A1KDM4EMEN1
SCHEMBL1385121 0.88 PARP1 (0.54) PARP1PARP2ALDH1A1KDM4EPOLB
SCHEMBL487963 0.80 ALDH1A1 (0.56) PARP1PARP2ALDH1A1KDM4EPOLB
SCHEMBL18108811 0.79 PARP1 (0.53) PARP1PARP2ALDH1A1KDM4EMEN1
SCHEMBL18040375 0.78 PARP1 (0.57) PARP1PARP2ALDH1A1KDM4EKMT2A
SCHEMBL16462030 0.75 ALDH1A1 (0.51) PARP1PARP2ALDH1A1KDM4EKMT2A
SCHEMBL1384426 0.75 PARP1 (0.50) PARP1PARP2ALDH1A1KDM4ESIGMAR1
SCHEMBL7739805 0.75 ERN1 (0.47) ALDH1A1KDM4EPOLBSIGMAR1KMT2A
SCHEMBL7737972 0.74 ERN1 (0.49) ALDH1A1KDM4EPOLBSIGMAR1KMT2A
SCHEMBL2228234 0.74 KDM4E (0.58) PARP1PARP2ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002020437-A2 BASIC COMPOUNDS CONTAINING TERTIARY AMIDES WITH ACTIVITY ON TACHYKININ RECEPTORS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2002-03-14 WO claimed
WO-2002020437-A2 BASIC COMPOUNDS CONTAINING TERTIARY AMIDES WITH ACTIVITY ON TACHYKININ RECEPTORS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2002-03-14 WO disclosed