SCHEMBL7526324

SCHEMBL7526324

COc1ccc2c(C(=O)C(=O)O)cn(C)c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
ABCG2 Q9UNQ0 2/20 0.48
NR4A2 P43354 2/20 0.43
SERPINE1 P05121 2/20 0.43
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
NQO2 P16083 1/20 0.42
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4003650 0.91 ABCG2 (0.57) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL5242703 0.88 ALDH1A1 (0.57) ALDH1A1ABCG2NR4A2KDM4EHPGD
SCHEMBL7503200 0.87 ALDH1A1 (0.54) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL5243737 0.84 NR4A2 (0.63) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL11392045 0.81 ALDH1A1 (0.59) ALDH1A1ABCG2KDM4EHPGDHSD17B10
SCHEMBL5241461 0.81 NR4A2 (0.54) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL29052011 0.80 HTT (0.61) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL4002802 0.79 SERPINE1 (0.47) ALDH1A1NR4A2SERPINE1KDM4EHPGD
SCHEMBL4406870 0.79 ABCG2 (0.60) ALDH1A1ABCG2NR4A2MTNR1AMTNR1B
SCHEMBL7522675 0.79 ALDH1A1 (0.44) ALDH1A1NR4A2SERPINE1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242409-A2 SUBSTITUTED BISINDOLYLMALEIMIDES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-25 EP disclosed
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2001046178-A2 SUBSTITUIERTE BISINDOLYMALEIMIDE F. HOFFMANN-LA ROCHE AG (CH) 2001-06-28 WO disclosed