SCHEMBL7526429

SCHEMBL7526429

Cn1c(=O)c2nc(-c3ccccc3)c(-c3ccccc3)nc2n(C)c1=O

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.78
ALDH1A1 P00352 6/20 0.78
HPGD P15428 3/20 0.78
GAA P10253 3/20 0.78
GLA P06280 1/20 0.78
ADORA2B P29275 3/20 0.55
ADORA2A P29274 2/20 0.55
HSD17B10 Q99714 2/20 0.52
CYP1A2 P05177 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
ADORA1 P30542 1/20 0.52
BLM P54132 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
LMNA P02545 2/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
HTT P42858 3/20 0.47
JAK2 O60674 1/20 0.47
PAX8 Q06710 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5447101 0.88 KDM4E (0.67) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL5441255 0.88 KDM4E (0.71) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL5452939 0.88 KDM4E (0.89) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL6314617 0.88 KDM4E (0.67) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL6314769 0.86 ALDH1A1 (0.64) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL5445201 0.83 ALDH1A1 (0.61) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL6315872 0.82 KDM4E (0.63) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL6321034 0.82 KDM4E (0.60) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL5447095 0.82 KDM4E (0.60) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL5449135 0.81 ALDH1A1 (0.58) KDM4EALDH1A1HPGDGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187615-A2 IMMUNOSURPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES K.U. Leuven Research & Development (BE) 2002-03-20 EP disclosed
WO-2000045800-A2 IMMUNOSURPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2000-08-10 WO disclosed
US-4038031-A REACTION WITH DIAZONIUM COMPOUND MILES LABORATORIES, INC. (US) 1977-07-26 US disclosed