SCHEMBL752801

SCHEMBL752801

C#Cc1ccc(-c2c[nH]c(C3CCCN3C(=O)CC(C)CNC(=O)OC)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.40
CYP2C9 P11712 5/20 0.38
KCNH2 Q12809 2/20 0.37
NR1I2 O75469 2/20 0.37
ABCB11 O95342 1/20 0.37
OPRK1 P41145 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP2D6 P10635 2/20 0.35
CPT1A P50416 8/20 0.34
CPT2 P23786 6/20 0.34
PRCP P42785 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16986624 0.85 CYP3A4 (0.38) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL750891 0.85 CYP3A4 (0.38) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL751612 0.84 CYP3A4 (0.56) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL2708006 0.81 CYP3A4 (0.61) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL205032 0.81 CYP3A4 (0.61) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL19388693 0.78 CYP3A4 (0.38) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL752193 0.78 CYP3A4 (0.32) CYP3A4CPT1A
SCHEMBL18534458 0.78 CYP3A4 (0.41) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL14331346 0.77 PRCP (0.35) CYP3A4CYP2C9CPT1ACPT2PRCP
SCHEMBL17527121 0.77 CPT1A (0.42) CYP3A4KCNH2CPT1ACPT2PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed