SCHEMBL752193

SCHEMBL752193

COC(=O)NCC(C)CC(=O)N1CCNCC1c1nc(-c2ccc(Br)cc2)c[nH]1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.32
DPP4 P27487 3/20 0.31
DPP7 Q9UHL4 2/20 0.31
CPT1A P50416 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL203743 0.81 CYP3A4 (0.51) CYP3A4
SCHEMBL752801 0.78 CYP3A4 (0.40) CYP3A4CPT1A
SCHEMBL18534458 0.76 CYP3A4 (0.41) CYP3A4CPT1A
SCHEMBL750891 0.75 CYP3A4 (0.38) CYP3A4CPT1A
SCHEMBL16986624 0.75 CYP3A4 (0.38) CYP3A4CPT1A
SCHEMBL17656270 0.74 CYP3A4 (0.49) CYP3A4
SCHEMBL18534351 0.72 KMT2A (0.38)
SCHEMBL748770 0.72 CYP3A4 (0.59) CYP3A4
SCHEMBL15349797 0.71 CYP3A4 (0.45) CYP3A4
SCHEMBL18534469 0.71 HCRTR1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596936-B Antiviral compounds GILEAD SCIENCES INC 2014-06-11 CN disclosed
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed