SCHEMBL7528052

SCHEMBL7528052

O=C(N[C@@H]1C2CCN(CC2)C1I)c1ccc(Sc2cnc(Cl)s2)s1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 16/20 0.43
CHRNB2 P17787 13/20 0.43
CHRNA4 P43681 13/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7063967 0.88 CHRNA7 (0.41) CHRNA7CHRNB2CHRNA4
SCHEMBL7524152 0.80 CHRNA7 (0.46) CHRNA7CHRNB2CHRNA4
SCHEMBL7061059 0.80 CHRNA7 (0.54) CHRNA7
SCHEMBL7063353 0.77 CHRNA7 (0.44) CHRNA7CHRNB2CHRNA4
SCHEMBL7063539 0.75 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL7062238 0.75 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL7063496 0.74 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL7063436 0.74 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL7061370 0.74 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL7061942 0.74 CHRNA7 (0.41) CHRNA7CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002017358-A2 QUINUCLIDINE-SUBSTITUTED HETEROARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO disclosed