SCHEMBL7528335

SCHEMBL7528335

Cc1cccc(C)c1N=C=O.Cc1ccccc1N=C=O.O=C=Nc1ccccc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.45
TRPA1 O75762 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
RAC1 P63000 1/20 0.34
PAK1 Q13153 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
GRIN2D O15399 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093597 0.93 CYP3A4 (0.47) CYP3A4TRPA1MEN1KMT2ACASP3
SCHEMBL75037 0.83 GABRA1 (0.43) CYP3A4TRPA1GABRA1GABRB2MEN1
SCHEMBL29648814 0.83 CYP3A4 (0.47) CYP3A4TRPA1MEN1KMT2ACASP3
SCHEMBL75112 0.83 CYP3A4 (0.47) CYP3A4TRPA1MEN1KMT2ACASP3
SCHEMBL7728938 0.79 KCNK3 (0.38) CYP3A4TRPA1MEN1KMT2ANOS3
SCHEMBL93287 0.78 CYP3A4 (0.64) CYP3A4TRPA1GABRA1GABRB2MEN1
SCHEMBL29541215 0.78 CYP3A4 (0.64) CYP3A4TRPA1GABRA1GABRB2MEN1
SCHEMBL3460968 0.77 CYP3A4 (0.66) CYP3A4TRPA1GABRA1GABRB2MEN1
SCHEMBL30520271 0.76 CYP3A4 (0.63) CYP3A4TRPA1GABRA1GABRB2MEN1
SCHEMBL20145 0.76 CYP3A4 (0.63) CYP3A4TRPA1GABRA1GABRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed