Iminostilbene

Iminostilbene

SCHEMBL75288

C1=Cc2ccccc2Nc2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 1.00
GAA P10253 5/20 1.00
NOX1 Q9Y5S8 4/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
BCHE P06276 3/20 0.43
ACHE P22303 3/20 0.43
POLB P06746 2/20 0.43
ALOX15 P16050 2/20 0.43
MAOA P21397 2/20 0.43
ALOX5 P09917 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ALOX12 P18054 1/20 0.43
CNR1 P21554 1/20 0.43
PTGS1 P23219 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2C P28335 1/20 0.43
PTGS2 P35354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iminostilbene SCHEMBL29926907 1.00 MAPT (1.00) MAPTGAANOX1MEN1KMT2A
Iminostilbene SCHEMBL5063042 0.97 MAPT (0.94) MAPTGAANOX1MEN1KMT2A
Iminostilbene SCHEMBL9685179 0.97 MAPT (0.94) MAPTGAANOX1MEN1KMT2A
SCHEMBL10449074 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL272082 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL10448842 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL19358 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL29870379 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL269763 0.82 MAPT (0.68) MAPTGAANOX1MEN1KMT2A
SCHEMBL1087950 0.81 GAA (0.68) MAPTGAANOX1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7416 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4406387-B1 AN ORGANIC ELECTRONIC DEVICE COMPRISING A SUBSTRATE, AN ANODE LAYER, A CATHODE LAYER, AT LEAST ONE FIRST EMISSION LAYER, AND A HOLE INJECTION LAYER, WHEREIN THE HOLE INJECTION LAYER COMPRISES A METAL COMPLEX OF FORMULA (I) AND A COMPOUND OF FORMULA (II), WHEREIN THE HOLE INJECTION LAYER IS ARRANGED BETWEEN THE ANODE LAYER AND THE AT LEAST ONE FIRST EMISSION LAYER NOVALED GMBH (DE) 2026-05-20 EP claimed
EP-4735585-A1 ENHANCING NEURONAL DIFFERENTIATION OF NEURAL PROGENITOR CELLS Novo Nordisk A/S (DK) 2026-05-06 EP claimed
US-12590297-B2 Differentiation method KONINKLIJKE NEDERLANDSE AKADEMIE VAN WETENSCHAPPEN (NL) 2026-03-31 US claimed
EP-4518635-B1 ORGANIC ELECTRONIC DEVICE COMPRISING A HOLE INJECTION LAYER, WHEREIN THE HOLE INJECTION LAYER COMPRISES A COMPOUND OF FORMULA (I) AND A COMPOUND OF FORMULA (III) NOVALED GMBH (DE) 2026-03-25 EP claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
EP-4344390-B1 ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING A RADIALENE OF FORMULA (I) AND A COMPOUND OF FORMULA (II), AND DISPLAY DEVICE COMPRISING THE ORGANIC ELECTROLUMINESCENT DEVICE NOVALED GMBH (DE) 2026-03-04 EP claimed
US-20260049268-A1 IN VITRO CELL CULTURE MUCUS SYSTEMS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2026-02-19 US claimed
US-20260043007-A1 METHOD FOR PRODUCING CARDIAC MUSCLES KYOTO UNIVERSITY (JP) 2026-02-12 US claimed
EP-4169084-B1 ORGANIC ELECTRONIC DEVICE COMPRISING A COMPOUND OF FORMULA (I), DISPLAY DEVICE COMPRISING THE ORGANIC ELECTRONIC DEVICE NOVALED GMBH (DE) 2026-01-28 EP claimed
US-12485126-B2 Combination for treating cancer INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2025-12-02 US claimed
US-4370324-A Method and composition for treating and preventing irritation of the eyes BERNSTEIN JOEL E (US) 1983-01-25 US claimed
WO-1983000086-A1 USE OF CALMODULIN BINDING DRUGS IN UTERUS TO PREVENT PREGNANCY UNIV GEORGIA RES FOUND (US) 1983-01-20 WO claimed
EP-0063525-A1 Dibenzazepine tetracyclic derivatives, process for their preparation and pharmaceutical compositions containing them CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 1982-10-27 EP claimed
EP-0053108-A1 VAGINAL CONTRACEPTIVES COMPRISING PSYCHOACTIVE DRUGS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1982-06-09 EP claimed
EP-0048023-A2 Composition for treating and preventing irritation of the eyes Bernstein, Joel E., M.D. (US) 1982-03-24 EP claimed
WO-1981003421-A1 USE OF PSYCHOACTIVE DRUGS AS VAGINAL CONTRACEPTIVES UNIV GEORGIA (US) 1981-12-10 WO claimed
US-4255329-A QUALITATIVE AND QUANTITATIVE ANALYSIS; SENSITIVITY; SPECTROPHOTOMERY SYVA COMPANY (US) 1981-03-10 US claimed
US-4249003-A Process for polycyclic amines AKTIEBOLAGET LEO (SE) 1981-02-03 US claimed
US-4124583-A 5-Substituted derivatives of 5H-dibenz (b,f)-azepine and method for obtaining the same DSO "PHARMACHIM" (BG) 1978-11-07 US claimed
US-4076812-A 10-Halogeno- or 10,11-dihalogeno derivatives of 5H-dibenz[b,f]azepine CIBA-GEIGY CORPORATION (US) 1978-02-28 US claimed