SCHEMBL7531986

SCHEMBL7531986

COC[C@H]1O[C@@H](n2cnc3c(Nc4cccc(F)c4)nc(C)nc32)[C@H](O)[C@@H]1O

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.61
ADORA1 P30542 1/20 0.61
NT5E P21589 1/20 0.51
ADORA2A P29274 1/20 0.49
DNPH1 O43598 1/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
GLA P06280 1/20 0.48
PMP22 Q01453 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531991 1.00 ADORA3 (0.61) ADORA3ADORA1NT5EADORA2ADNPH1
SCHEMBL7526418 0.91 ADORA3 (0.59) ADORA3ADORA1NT5EDNPH1ALDH1A1
SCHEMBL7526426 0.91 ADORA3 (0.59) ADORA3ADORA1NT5EDNPH1ALDH1A1
SCHEMBL7531045 0.90 ADORA3 (0.61) ADORA3ADORA1NT5EADORA2ADNPH1
SCHEMBL7531052 0.90 ADORA3 (0.61) ADORA3ADORA1NT5EADORA2ADNPH1
SCHEMBL7531536 0.90 ADORA3 (0.68) ADORA3ADORA1NT5EADORA2A
SCHEMBL7531527 0.90 ADORA3 (0.68) ADORA3ADORA1NT5EADORA2A
SCHEMBL8375864 0.89 ADORA3 (0.58) ADORA3ADORA1NT5EADORA2ADNPH1
SCHEMBL7526882 0.88 ADORA3 (0.79) ADORA3ADORA1NT5EADORA2A
SCHEMBL7527076 0.86 ADORA3 (0.55) ADORA3ADORA1NT5EADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901499-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2002-04-10 EP claimed
US-5998388-A N6-PHENYL-SUBSTITUTED GLAXO WELLCOME INC. (US) 1999-12-07 US claimed
EP-0901499-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2002-04-10 EP disclosed
US-5998388-A N6-PHENYL-SUBSTITUTED GLAXO WELLCOME INC. (US) 1999-12-07 US disclosed